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西咪替丁片的使用方法有什么呢?(西咪替丁片功效与作用)

发布时间2022-03-24 17:01:19  来源:粤迅康
【导读】西咪替丁片的使用方法有什么呢?:西咪替丁片用于治疗十二指肠溃疡、胃溃疡、反流性食管炎、应激性溃疡及卓-艾氏(Zollinger-Ellison)综合征。
西咪替丁片(泰胃美) ¥ 17.90元

规格:0.4g*10s

作用:临床主要用于:①各种酸相关性疾病:如十二指肠溃疡、胃溃疡、卓-艾综合征、上消化道出血、反流性食管炎、高酸性胃炎等。②据报道,可用于治疗带状疱疹和包括生殖器在内的其它疱疹性感染。

西咪替丁片为白色片或加有着色剂的淡蓝色或浅绿色片,或为薄膜衣片。那么,西咪替丁片的使用方法有什么呢?

西咪替丁片(泰胃美)

西咪替丁片用于治疗十二指肠溃疡、胃溃疡、反流性食管炎、应激性溃疡及卓-艾氏(Zollinger-Ellison)综合征。西咪替丁片口服后约60%~70%由肠道迅速吸收,西咪替丁片的血药浓度达峰时间(tmax)为45~90分钟。西咪替丁片口服生物利用度(F)约为70%,西咪替丁片对年轻人的吸收情况往往较老年人好。西咪替丁片的血浆蛋白结合率低。

西咪替丁片服用300mg平均峰浓度(Cmax)为1.44μg/ml,西咪替丁片可以抑制基础胃酸分泌50%达4~5小时。西咪替丁片广泛分布于全身组织(除脑以外),西咪替丁片在肝脏内代谢,主要经肾排泄。西咪替丁片24小时后口服量的约48%以原形自肾排出;10%从粪便排出。西咪替丁片可以经血液透析清除。西咪替丁片对肾功能正常时半衰期(t1/2)为2小时,西咪替丁片对肌酐清除率在20~50ml/分,西咪替丁片的半衰期(t1/2)为2.9小时,当<20ml/分时为3.7小时,西咪替丁片对肾功能不全时为5小时。西咪替丁片可经胎盘转运和从乳汁排出。西咪替丁片的使用方法是:

1.治疗十二指肠溃疡或病理性高分泌状态,一次0.2~0.4g(1-2片),一日4次,餐后及睡前服,或一次0.8g,睡前1次服。

2.预防溃疡复发,一次0.4g(2片),睡前服。

3.肾功能不全患者用量减为一次0.2g(1片),12小时1次。

4.老年患者用量酌减。

5.小儿:口服,一次按体重5~10mg/Kg,一日2~4次。

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