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儿童用 氢溴酸右美沙芬(中枢神经系统反应包括哪些)

发布时间2022-01-27 18:28:38  来源:粤迅康
【导读】氢溴酸右美沙芬片可以和其他中枢神经系统抑制药物合用吗?:氢溴酸右美沙芬片在进入体循环前通过肠壁、门脉及肝(有首过效应)。血浆中原型药物(右吗喃)浓度很低。
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<p>氢溴酸右美沙芬片每片含氢溴酸右美沙芬15毫克。辅料为淀粉、预胶化淀粉、蔗糖、硬脂酸镁。那么,氢溴酸右美沙芬片可以和其他中枢神经系统抑制药物合用吗?

氢溴酸右美沙芬片在进入体循环前通过肠壁、门脉及肝(有首过效应)。血浆中原型药物(右吗喃)浓度很低。有3-羟-甲氧吗啡烷、3-羟17-甲吗啡烷、3-羟吗啡烷三个主要代谢产物,并有较大的个体差异。单剂量给药和连续服用7天的代谢排泄基本相同。犬口服本品(20mg/kg)放射标记测定,70%为原型药物和三个主要代谢产物,血浆Cmax为2.5~5.0毫克当量/L(以右吗嘀计)Tmax为2~4h。

氢溴酸右美沙芬片为中枢性镇咳药,可抑制延脑咳嗽中枢而产生镇咳作用。其镇咳作用与可待因相等或稍强。一般治疗剂量不抑制呼吸,长期服用无成瘾性和耐受性。

氢溴酸右美沙芬片不宜与乙醇及其他中枢神经系统抑制药物并用,因可增强对中枢的抑制作用。

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