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宝诺达胞磷胆碱钠片(胞磷胆碱钠片是治什么的)

发布时间2021-12-02 11:01:13  来源:粤迅康
【导读】胞磷胆碱钠片的注意事项有什么呢?:胞磷胆碱钠片为白色或类白色片。胞磷胆碱钠片用于急性颅脑外伤和脑术后意识障碍。胞磷胆碱钠片口服:每日2次~3次,成人每次0.1g~0.2g(1/2-1片),儿童每次0.1g(1/2片)。
胞磷胆碱钠片(欣可来) ¥ 35.00元

规格:0.2g*12片/盒

作用:用于急性颅脑外伤和脑术后意识障碍。

胞磷胆碱钠片的主要成份会是:主要成分为胞磷胆碱钠。化学名:胆碱胞嘧啶核苷二磷酸酯单钠盐。分子式:C14H25N4(NaO)11P2。分子量:510.31。那么,胞磷胆碱钠片的注意事项有什么呢?

胞磷胆碱钠片(欣可来)

胞磷胆碱钠片为白色或类白色片。胞磷胆碱钠片用于急性颅脑外伤和脑术后意识障碍。胞磷胆碱钠片口服:每日2次~3次,成人每次0.1g~0.2g(1/2-1片),儿童每次0.1g(1/2片)。

胞磷胆碱钠片为核苷衍生物,胞磷胆碱钠片通过降低脑血管阻力,胞磷胆碱钠片具有增加脑血流而促进脑物质代谢,改善脑循环。胞磷胆碱钠片尚无口服给药的人体药代动力学资料。胞磷胆碱钠片的文献资料显示,胞磷胆碱钠片注射给药后血药浓度迅速下降,30分钟降至注入时的1/3,1-2小时基本稳定,胞磷胆碱钠片的分布以肝内最多,占10%,大部分于2小时内排人尿中。胞磷胆碱钠片较难通过血脑屏障,进入脑内的药物很少,仅占0.1%,但药物在脑内停留时间很长,胞磷胆碱钠片注射后3小时内药物浓度达峰值,并在24小时内保持不变,而且损伤脑比正常脑、受损半球比未受损半球的胞磷胆碱含量明显升高。

胞磷胆碱钠片动物实验显示,胞磷胆碱钠片口服则缓慢地完全吸收,胞磷胆碱钠片与静脉相比两者作用无显著差异。胞磷胆碱钠片口服给药能避免有害刺激,胞磷胆碱钠片增加低氧下动物存活时间。胞磷胆碱钠片的药物动力学研究表明,胞磷胆碱钠片口服给药,胞磷胆碱钠片可进入脑代谢,产生磷脂化作用而生效。胞磷胆碱钠片可增强脑干网状结构上行激活系统的机能,胞磷胆碱钠片具有增强锥体系统的机能,胞磷胆碱钠片可以改善运动麻痹,胞磷胆碱钠片对促进大脑功能的恢复和促进苏醒,有一定作用。

胞磷胆碱钠片的注意事项:脑出血急性期不宜大剂量应用。肌注一般不采用,若用时应经常更换注射部位。

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